Fatty alcohol esters
Medchemexpress LLC Cetrorelix Acetate | 145672-81-7 | 99.9% | 1491.09 | 1 MG
Cetrorelix Acetate is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist that inhibits the growth of the ES-2 cell line. It exhibits antiproliferative effects comparable to GnRH-I agonists. This product has a high purity of 99.9% and is supplied as a white to off-white solid. It requires specific storage conditions to maintain its stability, with powder stable for up to 2 years at -80°C and solutions for up to 6 months at -80°C.
- Potent GnRH receptor antagonist
- Inhibits ES-2 cell line growth
- Comparable antiproliferative effects to GnRH-I agonists
- High purity
- Stable under specific storage conditions
Medchemexpress LLC Mait-203 (acetate) | 99.1% | 2577.90 | 1 MG
MAIT-203 acetate is a cyclopentyalanin-derived peptidomimetic that potently inhibits the interaction of adenomatous polyposis coli (APC) and Asef (RhoGEF4). It binds APC-ARM with a Ki value of 0.015 μM and a Kd value of 0.036 μΜ, significantly repressing the migration and invasion of colorectal cancer cells.
- Reduces Asef-APC interaction in a dose-dependent manner in HEK293T cells.
- Attenuates SW480 and HCT116 cell migration.
- Decreases the amount of active CDC42 in SW480 cells.
Medchemexpress LLC Histrelin acetate | 220810-26-4 | 99.9% | 1323.50 (free base) | 10 MG
Histrelin acetate is a GnRH analogue and a GnRH Receptor agonist. It increases serum luteinising hormone (LH), follicle stimulating hormone (FSH), and testosterone levels. It can be used in the research of prostate cancer and endometriosis.
- Stimulates the release of vasopressin (VP) and oxytocin (OT) from isolated rat hypothalamo-neurohypophysial explants.
- Rescues circulating LH concentrations in Csfmop/Csfmop mice.
- Reduces the number of endometrial glands, atrophying the stroma in rabbits.
Medchemexpress LLC Glp-1(7-37) acetate | 1450806-98-0 | 99.59% | 3355.67 (free base) | 10 MG
GLP-1(7-37) acetate is an intestinal insulinotropic hormone that augments glucose induced insulin secretion and is for research use only.
- Augments glucose induced insulin secretion
- Solid appearance
- White to off-white color
- Sequence: His-Ala-Glu-Gly-Thr-Phe-Thr-Ser-Asp-Val-Ser-Ser-Tyr-Leu-Glu-Gly-Gln-Ala-Ala-Lys-Glu-Phe-Ile-Ala-Trp-Leu-Val-Lys-Gly-Gr-Gly
- Soluble in H2O: 50 mg/mL (ultrasonic and adjust pH to 1 with HCl)
- Soluble in PBS: 2 mg/mL (clear solution; need ultrasonic)
Medchemexpress LLC Retinyl acetate | 127-47-9 | MFCD00019413 | 328.49 | 50 MG
Retinyl acetate is a synthetic acetate ester derived from retinol, demonstrating potential antineoplastic and chemopreventive activities. It has been shown to inhibit the proliferation of tumor cells and is suitable for various in vitro and in vivo studies.
- Inhibits proliferation of tumor cells, such as melanoma cell lines B16 and S91
- Inhibits DMBA-induced mammary carcinogenesis in Sprague-Dawley rats
- Appears as a solid, off-white to light yellow in color
- Soluble in DMSO and corn oil for experimental applications
Medchemexpress LLC Anecortave acetate 10mg | 7753-60-8 | 386.5 g/mol | C23H30O5 | 10 MG
Anecortave acetate is a steroidal angiostatic agent used in research on ocular neovascularization and age-related macular degeneration. It is supplied as a high-purity research reagent with supporting analytical documentation and handling guidance.
- High reported purity, suitable for research use.
- Molecular weight 386.5 g/mol and formula C23H30O5.
- Available in a 10 mg research package.
- Analytical documentation available, including COA, HNMR, and LCMS.
- Used in studies of angiogenesis and retinal neovascular disorders.
Medchemexpress LLC Lefamulin acetate | 1350636-82-6 | 99.7% | 567.78 | 1 ML
Lefamulin acetate is an orally active antibiotic that inhibits protein synthesis by binding to the peptidyl transferase center of the 50S bacterial ribosome. It also demonstrates anti-inflammatory activity and is utilized in research pertaining to bacterial infections, such as bacterial pneumonia.
- Inhibits protein synthesis by binding to 50S bacterial ribosome.
- Exhibits anti-inflammatory activity.
- Effective against C. trachomatis, N. gonorrhoeae, and M. genitalium.
- Potent activity against M. pneumoniae strains.
- Shows antibacterial effect in S. pneumoniae or S. aureus challenged lung infection mice.
- Reduces BALF neutrophil cell counts and levels of pro-inflammatory cytokines and chemokines in LPS-induced lung neutrophilia mouse model.
Medchemexpress LLC Sifuvirtide acetate | 99.8% | 4727.98 | 1 MG
Sifuvirtide acetate is a potent HIV fusion inhibitor. It inhibits HIV-1 mediated cell fusion in a dose-dependent manner and is highly potent against infection by primary and laboratory-adapted HIV-1 isolates of multiple genotypes. Sifuvirtide acetate can be used in the research of anti-HIV drugs.
- Potent HIV fusion inhibitor
- Inhibits HIV-1 mediated cell fusion in a dose-dependent manner
- Highly potent against infection by primary and laboratory-adapted HIV-1 isolates of multiple genotypes
- Can be used in the research of anti-HIV drugs
Medchemexpress LLC NN1213 acetate | 99.7% | 4553.10 (free base) | 10 MG
NN1213 acetate is a long-acting human amylin peptide analog and a selective amylin receptor agonist. It has EC50 values of 0.177 nM for hAMY3R and 0.262 nM for rAMY3R. This compound significantly reduces food intake and fat mass, leading to body weight reduction in diet-induced obese rats, making it suitable for obesity research.
- Selective amylin receptor agonist
- EC50 values of 0.177 nM for hAMY3R and 0.262 nM for rAMY3R
- Produces dose-dependent body weight loss in diet-induced obese rats
- Reduces food intake in rats and beagle dogs
- Decreases body weight and food intake in diet-induced obese rats
Medchemexpress LLC Cggk acetate | 96.8% | 363.43 | 10 MG
CGGK acetate is a control peptide for CAQK peptide. This peptide is provided as a solid, white to off-white appearance with a purity of 96.78%. It is suitable for various research applications.
- For research use only
- Ships at room temperature in continental US
- Store sealed, away from moisture
- Soluble in DMSO (≥ 100 mg/mL)
Medchemexpress LLC α-Amyrin acetate | 863-76-3 | 1 MG
α-Amyrin acetate is a pentacyclic triterpenoid compound with oral activity. It inhibits cancer cell proliferation, induces apoptosis, and reduces blood glucose levels. This compound is used for research in cancer and metabolic diseases, such as breast cancer and diabetes.
- Inhibits proliferation and colony formation in MDA-MB-231 cells.
- Induces apoptosis and increases caspase-3 activity in MDA-MB-231 cells.
- Promotes cleavage of Poly polymerase, increases E-cadherin, and inhibits vimentin and phosphorylated extracellular signal-regulated activation in MDA-MB-231 cells.
- Reduces blood glucose levels in diabetic rats.
Medchemexpress LLC JMV 449 acetate | 141863-45-8 | 99.7% | 807.03 | 1 MG
JMV 449 acetate is a potent neurotensin receptor agonist. It exhibits an IC50 of 0.15 nM for inhibiting 125I-neurotensin binding to neonatal mouse brain and an EC50 of 1.9 nM in contracting the guinea-pig ileum. This product also demonstrates highly potent and long-lasting hypothermic and analgesic effects in mice.
- Potent neurotensin receptor agonist
- IC50 of 0.15 nM for inhibition of 125I-neurotensin binding
- EC50 of 1.9 nM in contracting guinea-pig ileum
- Highly potent and long-lasting hypothermic effects
- Highly potent and long-lasting analgesic effects in mice
- White to off-white solid appearance
- Soluble in H2O at 100 mg/mL (requires ultrasonic)
Medchemexpress LLC LSD (acetate) | 945245-76-1 | 98.0% | 1009.20 | 10 MG
LSD acetate is a peptide utilized in targeted therapy and diagnosis research for tumor lymphatics. It specifically recognizes the lymphatics of C8161 melanoma, without binding to normal tissue lymphatics or tumor blood vessels. When conjugated with a proapoptotic peptide, it can effectively reduce the number of tumor lymphatics.
- Recognizes C8161 melanoma lymphatics
- Does not bind to normal tissue lymphatics or tumor blood vessels
- Reduces tumor lymphatics when conjugated with proapoptotic peptides
- Suitable for targeted therapy research
- Suitable for diagnosis of tumor lymphatics
TARGETMOL CHEMICALS INC Terlipressin Acetate 25MG
Also available in 5 mg, 10 mg, 50 mg, 100 mg, 200 mg and bulk. Please contact Fisher for quotes. Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelial cells (IEC-6).Terlipressin acetate exerts anti-inflammatory and anti-oxidative effects. Terlipressin acetate has the potential for hepatorenal syndrome and norepinephrine-resistant septic shock research. Purity 99.69%
Medchemexpress LLC Sgnrh-A acetate | 99.9% | 1342.50 | 10 MG
sGnRH-A acetate is a salmon gonadotropin-releasing hormone (GnRH) analogue. It stimulates growth hormone secretion and can be used as an inducer of ovulation by artificial insemination.